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生物活性小分子专题生物活性小分子肿瘤是现代一种严重威胁人类健康的常见病和多发病,研制靶向性抗肿瘤药物成为了肿瘤治疗研究中的热点领域。小分子抑制剂能特异性结合到靶蛋白上, 选择性地阻断肿瘤细胞的过度增生, 从而有效控制和治疗疾病。 阿拉丁生物活性小分子是一类用于实验研究的PI3K/Akt/mTOR,血管内皮生长因子受体(VEGFR),JAK,细胞凋亡(Apoptosis),MAPK,HDAC和蛋白酶体(Proteasome)等上百个信号通路的高特异性小分子抑制剂。小分子抑制剂推荐-产品列表产品货号产品名称规格CAS价格/RMBA124776-1g阿替洛尔98%,powder29122-68-7629.00 A124880-1gAripiprazole99%129722-12-9519.00 A129250-10mgAzatadine dimaleate98%3978-86-7399.00 A129255-10mgAzilsartan99%147403-03-0479.00 A129323-5mgAfatinib99%439081-18-2689.00 A129429-1gAcemetacin98%53164-05-9212.82 A129498-5mgAZD198198%802904-66-1699.00 B129216-1gBenztropine mesylate98%132-17-2319.00 B129218-10mgBepotastine Besilate98%190786-44-8418.99 B129286-5gBufexamac98.0%(HPLC)2438-72-4399.00 B129734-10mgBRL-5444398%57477-39-1689.00 B129764-10mgBrivanib Alaninate (BMS-582664)95%649735-63-72199.00 B129826-10mgBrinzolamide98%138890-62-7299.00 B129864-5gBupivacaine HCl98%18010-40-7499.00 B129898-10mgBIBR 153298%321674-73-1799.00 C124969-1gCapecitabine99%154361-50-9899.00 C126883-1g氯氮平98%(GC)5786-21-0768.00 C127224-10mgCYT38798%1056634-68-41199.00 C129233-5g马来酸氯苯那敏99%113-92-8189.00 C129678-1g西洛他唑99%73963-72-1499.00 C129678-250mg西洛他唑99%73963-72-1219.00 C129746-1gClarithromycin98%81103-11-9169.00 D125392-5mgDelafloxacin98%189279-58-11399.00 D129347-5mgDacomitinib (PF299804, PF299)99%1110813-31-42099.00 D129639-1gDapoxetine hydrochloride98% (HPLC)129938-20-1699.00 D129790-50mgDidanosine98% (HPLC)69655-05-6259.00 D129813-5mgDexmedetomidine HCl98%145108-58-3499.00 D129815-50mgDetomidine HCl98%90038-01-0329.00 D129847-1gDacarbazine98%4342-03-4659.00 D129948-1gDonepezil HCl98%120011-70-3699.00 E105515-1g雌酮98.0%(GC)53-16-7143.10 E125682-10mgEPZ00568798%1396772-26-12499.00 E129310-100mgErlotinib HCl (OSI-744)99%183319-69-9699.00 E129317-5gEtodolac98%41340-25-4529.00 E129454-10mgTofacitinib (CP-690550) Citrate99%540737-29-9999.00 E129603-10mgGabapentin HCl98%60142-95-2489.00 F126912-10mgFenretinide98%65646-68-6359.00 F129242-5gFamotidine99%76824-35-6629.00 F129526-1gFlunarizine 2HCl99%30484-77-6186.32 F129671-1gFluvoxamine maleate98%61718-82-9469.23 F129812-10mgFormoterol Hemifumarate99%43229-80-7559.00 I125935-50mgIndacaterol99%312753-06-3799.00 I129263-1gIrbesartan98%138402-11-6579.00 I129957-1gIrsogladine98%57381-26-7869.00 J129258-10mgJNJ-777712098% (HPLC)459168-41-3799.00 K129289-1g酮咯酸氨丁三醇99%74103-07-4185.00 K129331-5gKetoprofen98%(HPLC)22071-15-4269.00 K129656-10mgKPT-18598%1333151-73-7659.00 K129737-1g酮康唑 98%65277-42-199.00 L125568-10mgLaropiprant99%571170-77-91629.00 L129223-100mgLoratadine98%79794-75-5429.00 L129227-1gLosartan potassium99%124750-99-8259.00 L129237-10mgLafutidine99%118288-08-7499.00 L129324-1gLisinopril Dihydrate98%83915-83-7829.00 L129338-100mg二对甲苯磺酸拉帕替尼(GW-572016)98%388082-77-71299.00 L129338-25mg二对甲苯磺酸拉帕替尼(GW-572016)98%388082-77-7499.00 L129341-250mgLornoxicam98% (HPLC)70374-39-9299.00 L129452-5gLevosulpiride98%23672-07-3519.00 L129465-5gLoperamide HCl98%34552-83-5558.00 L129522-50mgLacidipine98%103890-78-4289.00 L129555-1gLamotrigine98%84057-84-1649.00 L129692-10mgLY31076295%192927-92-7859.00 M125524-5mgMacitentan97%441798-33-0448.00 M125894-5mgM34497%251456-60-7448.00 M126151-5mgMocetinostat (MGCD0103)98%726169-73-9639.00 M126688-10mgMirabegron99%223673-61-81999.00 M126688-5mgMirabegron99%223673-61-81098.00 M126795-10mgMotesanib98%453562-69-1299.00 M126858-50mg6-巯基嘌呤 (6-MP)99%50-44-2309.00 M126981-25mgMasitinib (AB1010)98%790299-79-5899.00 M126999-1gMifepristone98%84371-65-3769.00 M127026-100mgMedetomidine98%86347-14-01842.00 M127205-5mgMK-824598%1030612-90-81699.00 M127991-5mgSuvorexant (MK-4305)98%1030377-33-3599.00 M129243-5mgMLN970898%1201902-80-81180.00 M129328-10mgMoexipril HCl98%82586-52-5529.00 M129409-1gMedroxyprogesterone acetate98%71-58-9289.00 M129573-50mgMitiglinide Calcium99%145525-41-3695.00 M129577-10mgML133 HCl98%1222781-70-5699.00 M129577-5mgML133 HCl98%1222781-70-5499.00 M129587-100mgMilrinone99%78415-72-2659.00 M129673-10mgMosapride Citrate98%112885-42-4349.00 M129673-50mgMosapride Citrate98%112885-42-41190.00 M129736-5mgMotesanib Diphosphate (AMG-706)98%857876-30-31190.00 M129842-10mgMizoribine98%50924-49-7299.00 M129842-50mgMizoribine98%50924-49-7899.00 M129859-50mgMildronate dihydrate98%86426-17-7629.00 M129861-50mgMoxifloxacin HCl99%186826-86-8599.00 M129872-10mgMozavaptan99%137975-06-51599.00 N126810-5mgNVP-ADW74299%475488-23-41099.00 N126962-5mgNVP-AUY92298%747412-49-31975.00 N129229-5gNizatidine98%76963-41-2299.00 N129262-10mgNafamostat Mesylate98%82956-11-4189.00 N129358-10mgNSC 40502098%7497-07-6699.00 N129506-1gNimodipine98%66085-59-4849.00 N129506-250mgNimodipine98%66085-59-4299.00 N129566-1gNicorandil98%(HPLC)65141-46-01499.00 N129604-50mgNefiracetam98%77191-36-7329.00 N129630-10mgNaratriptan hydrochloride98%143388-64-1449.00 N129630-50mgNaratriptan hydrochloride98%143388-64-11899.00 N129725-5mgNintedanib (BIBF 1120)98%656247-17-5869.00 N129741-10mgNU702698%154447-35-5529.00 N129779-100mgNevirapine98%(HPLC)129618-40-2389.00 N129779-500mgNevirapine98%(HPLC)129618-40-21599.00 N129805-5gNaftopidil98.0%57149-07-2749.00 N129985-10mgNU602798%220036-08-8999.00 O126519-1gOlanzapine99%132539-06-1678.00 O127017-10mgOC00045998%851723-84-7799.00 O127383-5mgObatoclax Mesylate97%803712-79-0999.00 O127572-5mgONX-0914 (PR-957)98%960374-59-8999.00 O129301-10mgOlmesartan Medoxomil98%144689-63-4799.00 O129301-50mgOlmesartan Medoxomil98%144689-63-42799.00 O129581-10mgOmecamtiv mecarbil (CK-1827452)98%873697-71-31899.00 O129581-5mgOmecamtiv mecarbil (CK-1827452)98%873697-71-31190.00 O129679-1gOndansetron Hydrochloride Dihydrate98% (HPLC)103639-04-9599.00 O129694-10mgOndansetron99%99614-02-5469.00 O129837-10mgOrg 2756998%868273-06-7799.00 O129871-10mgOzagrel98%82571-53-7599.00 O129945-1gOxybutynin98%5633-20-5699.00 O129950-5gOtilonium Bromide98%26095-59-0279.00 O129984-5gOrphenadrine Citrate95%4682-36-4319.00 P125212-10mgPNU-12059698% (HPLC)501925-31-1499.00 P125444-5mgPelitinib98%257933-82-7899.00 P125494-5mgPD032590199%391210-10-9569.00 P125813-10mgPomalidomide99%19171-19-8599.00 P125813-50mgPomalidomide99%19171-19-81980.00 P125823-10mgPQ 40199%196868-63-0969.00 P125865-5mgPD17307499%219580-11-7459.00 P126147-5mgPF-56227198%717907-75-0899.00 P126351-10mgPCI-3405198%950762-95-51099.00 P126419-10mgPP12198%1092788-83-4799.00 P126620-10mgPD9805998%167869-21-8869.00 P126755-10mgPitolisant98%362665-56-3989.00 P127355-10mgAtaluren (PTC124)99%775304-57-9499.00 P127387-10mgPSI-613098%817204-33-42699.00 P127387-5mgPSI-613098%817204-33-41699.00 P127550-10mgPonatinib (AP24534)99%943319-70-8699.00 P127795-5mgPHA-79388795%718630-59-21099.00 P127910-10mgPracinostat (SB939)98%929016-96-61999.00 P127910-5mgPracinostat (SB939)98%929016-96-61199.00 P127989-5mgPF-0445784598%1020315-31-41899.00 P128026-10mgPlerixafor98%110078-46-1999.00 P129261-10mgPemirolast potassium99%100299-08-9499.00 P129294-1gPiroxicam98%(HPLC)36322-90-4239.00 P129306-10mgPAC-198%315183-21-2589.00 P129384-10mgPD153035 HCl98%(HPLC)183322-45-4669.00 P129412-5g孕烯醇酮98%(GC)145-13-1179.00 P129434-10mgPramipexole99%104632-26-0299.00 P129447-10mgPD16839398%194423-15-91299.00 P129535-25g苯妥英99%57-41-0119.00 P129662-10mgPrucalopride99%179474-81-81198.00 P129680-10mgPimobendan99%74150-27-91590.00 P129680-5mgPimobendan99%74150-27-91098.00 P129711-1gParoxetine hydrochloride hemihydrate98% (HPLC)110429-35-1779.00 P129722-25mgPazopanib HCl (GW786034 HCl)98%635702-64-6759.00 P129744-100mgPalonosetron HCl99%135729-62-3599.00 P129781-10mgPluriSIn #1 (NSC 14613)98%91396-88-2699.00 P129811-5mgPF-0056227197%939791-38-51699.00 P129841-50mgPemetrexed99%150399-23-8339.00 P129843-1gPhenoxybenzamine HCl98%63-92-3297.00 P129846-10mgPlerixafor 8HCl (AMD3100 8HCl)99%155148-31-5419.00 P129846-5mgPlerixafor 8HCl (AMD3100 8HCl)99%155148-31-5259.00 P129854-50mgProcarbazine HCl98%366-70-1289.00 P129908-5mgPRT062607 (P505-15, BIIB057) HCl98%1370261-97-41119.00 P129961-10mgPifithrin-α (PFTα)97%63208-82-2869.00 P129976-25mgPancuronium dibromide99%15500-66-0829.00 P140269-250mgPemetrexed disodium hydrate99%357166-30-4349.00 Q127558-5mgQuizartinib (AC220)99%950769-58-12593.00 R125051-10mgRamelteon99%196597-26-91999.00 R125138-10mgRivaroxaban99%366789-02-8899.00 R125195-10mgR-147999%478182-28-42619.00 R125421-5mgRITA (NSC 652287)98%213261-59-7989.00 R126180-250mgRacecadotril98%81110-73-8249.00 R126338-5mgRuxolitinib (INCB018424)99%941678-49-5989.00 R126531-10mgRKI-144798%1342278-01-6889.00 R126586-10mgRitonavir98%155213-67-5589.00 R126586-50mgRitonavir98%155213-67-52419.00 R126814-10mgRG10898%48208-26-0149.00 R127644-10mgRisperidone99%106266-06-2268.00 R127804-5mgRegorafenib (BAY 73-4506)99%755037-03-7479.00 R129220-100mgRosuvastatin Calcium99%147098-20-22939.00 R129220-25mgRosuvastatin Calcium99%147098-20-2839.00 R129246-1g盐酸罗沙替丁醋酸酯99%93793-83-0829.00 R129396-100mgRaloxifene HCl98%82640-04-8479.00 R129396-25mgRaloxifene HCl98%82640-04-8169.00 R129533-1gRiluzole98%1744-22-5319.00 R129561-50mgRepaglinide99%135062-02-1699.00 R129638-10mgRizatriptan Benzoate98%(HPLC)145202-66-0319.00 R129674-10mgRolipram97%61413-54-5219.00 R129756-100mgRosiglitazone maleate99%155141-29-0699.00 R129756-25mgRosiglitazone maleate99%155141-29-0238.00 R129769-25mgRosiglitazone HCl99%302543-62-01999.00 R129769-5mgRosiglitazone HCl99%302543-62-0999.00 R129802-10mgRaltegravir (MK-0518)97%518048-05-01379.00 R129802-5mgRaltegravir (MK-0518)97%518048-05-0749.00 R129910-10mgR406 (free base)99%841290-80-01699.00 R129955-10mgRocuronium Bromide98%119302-91-9189.00 S125282-10mgSafinamide98%133865-89-1319.00 S125282-50mgSafinamide98%133865-89-11339.00 S125519-5mgSemagacestat (LY450139)98%425386-60-31299.00 S125580-25mgSelumetinib (AZD6244)99%606143-52-6289.00 S126595-5mgSilodosin99%160970-54-7499.00 S129544-500mgClopidogrel Bisulfate98%120202-66-6489.00 S129663-100mgSildenafil Citrate98% (HPLC)171599-83-01199.00 S129663-25mgSildenafil Citrate98% (HPLC)171599-83-0399.00 S129681-50mgSumatriptan Succinate98% (HPLC)103628-48-4369.00 S129783-1gStavudine (d4T)98%3056-17-5689.00 S129877-10mgSafinamide Mesylate98% (HPLC)202825-46-51099.00 S129877-5mgSafinamide Mesylate98% (HPLC)202825-46-5689.00 S129890-5mgSRT172098%1001645-58-4999.00 T125146-10mgTenovin-198%380315-80-0549.00 T125285-10mgTolcapone99%134308-13-7369.00 T125285-50mgTolcapone99%134308-13-7999.00 T125988-10mgSMI-4a98%438190-29-5679.00 T126745-10mgToceranib98%356068-94-5999.00 T126775-5mgTelaprevir98%402957-28-2899.00 T126856-1gThalidomide98%50-35-1499.00 T127425-250mgTemozolomide98% (HPLC)85622-93-1469.00 T127446-5mgTrelagliptin98%865759-25-71319.00 T129239-1gTelmisartan98%144701-48-4679.00 T129468-5gTrimebutine98%39133-31-8369.00 T129665-5mgTrichostatin A98%58880-19-61899.00 T129819-5mgTAE684 (NVP-TAE684)98%761439-42-3969.00 T129870-10mgTolvaptan98%150683-30-0869.00 T129870-50mgTolvaptan98%150683-30-02999.00 T129936-100mgTrospium chloride99%10405-02-41999.00 T129936-25mg

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