Petesicatib _Cathepsin 抑制剂 - MedChemExpress

1、Hotline: 400-820-3792Inhibitors Agonists Screening Librarieswww.MedChemEPetesicatibCat. No.: HY-109069CAS No.: 1252637-35-6分式: CHFNOS分量: 603.54作靶点: Cathepsin作通路: Metabolic Enzyme/Protease储存式: Powder -20C 3 years4C 2 yearsIn solvent -80C 6 months-20C 1 month溶解性数据体外实验 DMSO : 125 mg/mL (207.11 mM; Need

2、 ultrasonic)Mass Solvent1 mg 5 mg 10 mg Concentration制备储备液1 mM 1.6569 mL 8.2845 mL 16.5689 mL5 mM 0.3314 mL 1.6569 mL 3.3138 mL10 mM 0.1657 mL 0.8284 mL 1.6569 mL请根据产品在不同溶剂中的溶解度，选择合适的溶剂配制储备液，并请注意储备液的保存式和期限。体内实验 请根据您的实验动物和给药式选择适当的溶解案，配制前请先配制澄清的储备液，再依次添加助溶剂(为保证实验结果的可靠性，体内实验的作液，建议您现现配，当天使；澄清的储备液可以根据储存条

3、件，适当保存；以下溶剂前的百分 指该溶剂在您配制终溶液中的体积占)：1. 请依序添加每种溶剂： 10% DMSO 40% PEG300 5% Tween-80 45% salineSolubility: 2.08 mg/mL (3.45 mM); Clear solution2. 请依序添加每种溶剂： 10% DMSO 90% (20% SBE-CD in saline)Solubility: 2.08 mg/mL (3.45 mM); Clear solution3. 请依序添加每种溶剂： 10% DMSO 90% corn oilSolubility: 2.08 mg/mL (3.45 m

4、M); Clear solution1/2 Master of Small Molecules 您边的抑制剂师www.MedChemEBIOLOGICAL ACTIVITY物活性 Petesicatib种 cathepsin S 抑制剂，可于免疫疾病研究 1。IC50 & Target Cathepsin S 1体外研究 Petesicatib (Example 238) is a cathepsin S inhibitor, used in research of immune diseases 1.REFERENCES1. Rubn Alvarez Snchez, et al. Novel proline derivatives. US20100267722A1McePdfHeightCaution: Product has not been fully validated for medical applications.For research use only.Tel: 400-820-3792;Fax