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综述含哌嗪化合物作为受体配体的研究进展ADVANCEINPIPERAZINECONTAININGCOMPOUNDSASRECEPTORLIGANDSA1A0A1A0A2A3A4A3A4A5A6A7A8A9A10A11A12A13A14A15A16A17A18A19A18A20A21A22A23A24A25A26A27A28A29A30A31A32A33A34A35A36A37A38A39A40A41A42A30A43A44A45A46A47A48A49A50A51A52MC4RA53A54A55A56A57A52DAA53A50A51A54A50A51A545A58A59A57A525HTA53A50A51A60A51A61A62A63A64A65A66A67A68A69A70A25A71A72A73A74A75A71A72A73A74A28A39A40A41A76A42A30A43A44A45A77A78A64A50A51A60A51A79A80A81A82A64A83A43A84A85A86A87A88A89A67A68A90A91A64A84A92A93A94A95A96A86A97A98A67A68A64A99A100A101A102A86A103A80A104A105A104A55A64A106A107A85A108A54A109A110A111A112A113A85A48A114A64A39A40A41A109A43A115A116A117A118A25A119A120A121A119A120A121A122A122A122A40A41A123A46A47A48A49A50A51A123A55A56A57A50A51A1235A58A59A57A50A51A123A124A125A126A127A109A123A124A128A129A40A41A130A87A109A43A42A113A67A68A131A132A115A64A96A76A133A134A130A42A30A43A86A79A802A135A136A57A64A137A138A139A140A86A141A142A116A143A86A144A64A145A102A146A80A147A148A149A150A109A43A64A151A42A85A48A86A152A153A55A135A154A155A156A157A158A155A86A159A108A109A43A64A83A43A84A85A25A40A41A130A81A82A160A161A116A162A55A109A43A163A158A131A86A164A165A166A64A39A40A41A109A43A167A8070A55A168A86A169A170A171A81A82A64A83A43A84A85A25A172A173A105A86A67A68A174A175MC4RA54DAA545HTA54A50A51A54P2X7A50A51A54TRPV1A50A51A61A146A139A87A176A177A109A54A178A179A180A181A138A139A182A183A52ERECTILEDYSFUNCTIONA86EDA53A109A43A54A124A125A126A184A132A109A54A185A186A109A61A64A44A115A187A188A25A39A40A41A64A42A30A43A44A45A77A78A64A50A51A60A51A170A45A189A163A84A92A64A67A68A93A94A25A190A116A31A32A33A191A192A193A194A80A195A40A41A76A42A30A43A44A45A50A51A60A51A64A196A51A197A198A199A200A86A201A34A29A37A172A202A173A105A39A40A41A64A42A30A43A44A45A50A51A60A51A64A65A66A67A68A203A198A251MC4R配体11MC4RA204A205A206A205A206MC4RA207A208A209A210A211A212A213A214A215EDA216A217A218A219A220A221A222A223A224A225A226A227A228A229A230DA231A232A233A234A235PCLDPHEA236A237D1,2,3,4A238A2393A240A241A242A235DTICA236A243A244A245A246A247A248A249A226A227A250A251A2521A253A254A255A126A0A1A2A3A4A5A6A7A8A5A255A9A10A11A55A204A12A2A3A205A13A14A254A15A161A21A192A17A18A19CLA121FA209A20A8A22A23A24A25A26A27A2552A177A28A29A30A31A32A33A34A208A35A36A33A37A38A393A177MC4RA213A49A40A41A42A432A44A45A46A47A48A50A28A51A52A53A35A36DTICA218A54A56A57A58A59A221A60A61A62A63A64A65A66A67A68A69A70A71A72A7312MC4RA74A75A76A75A76MC4RA228A77A78A79A80A81A82A83A84A85A86A87A88CACHEXIAA89A110A90A91A92A93A94A185A95A96A97A98A99A100A101A102A1034A111A104A105MC4RA106A107A108A236A109A112A113A114A115A116A103A117A118A119A120A107A122A108A123A124A125A127A128A129MC4RA130A131A132A133A134A135A136A137A138A139A140A141A142A143A144A145A146A147A148A2463A149MC4RA150A151A130A131A132A152A153A145A154A155A156A157A158A159A160A161A162A163A149A251A164A165A166A167A168A1695A170A171A172A173A174A175A176A178A179A180A181A182A183A249A184A206A1864A187A188A189A190A191A193A194A195A196A197A198A199A200A201A2026A203IC5084NMOLL1A207A210A211A212A214A215A216A217A219A220A222A223A224A225A226A227A229A230A225A231A232A229A233A2345A235A2371MC4RA238A239FIG1MC4RLIGANDSA240A241A242MC4RA238A239A243A244A245A247A248A242MC4RA238A239A250A252A253A254A255A15A34A75A0A1A2A34A78A3A4A255A5A1A6A7A40A8A9A21A10A56A55A11A85A12A13A178A85A14A16A17A18A17A19A20A22A23A24A25A26A55A27A157A28A158A29A30A31A32A33A212D2家族多巴胺受体配体21A35A36A37D2A38A39A41A39A39A41D2A42A43A44A45A46A47A48A49A50A51A52A53A54A57A58A59A137A60A61A62A63A64A65A50A66A67A68A45A46A47A48A49A69A251A70A71A98A72A73OLANZAPINEA74A76A77A79A80A81ZIPRASIDONEA69A82A83A66A84A73ARIPIPRAZOLEA74A86A87A177D2A42A43A88A89A64A199A50A90A91A92A59PENJIEVIA866A62A63A93A94A95A105A96A105A66A67A177D2A42A43A50A97A99A100A101A177A102A103A104A106A59A193A107A97A108A139A109A110A111A112A99A113A1045HT1AA915HT2AA42A43A114A88A115A116A117A86A50A90A91A92A73KI100NMOLL1A74A69A104D2A42A43A114A88A118A90A91A92A73KI70NMOLL1A74A59A104A106A102A119A139A109A73IA74A101A103A112A50A66A67A120N1A208A177A121A122A123A124A182A125A126A105A50A127A128A53A54A129A73IIA74A130A43A50A121A122A131A102A177A132A182A125A76A133A182A125A76A134A182A125A76A135A182A125A183A136A50A138A140A129A73A141A74A192A105A66A67A131A102A50A192A120A177A96A142A182A125A143A144A182A125A126A105A50A145A146A127A128A53A54A59A110A111A97A108A147A148A100A149A150A65A151A152A153A112A99A113A154A155A156A105A159A5922A160A161A162D3A163A164A165A164A164A165A166A167A168A169A170A171D3A172A173A174A175A176A179A180A181A184A185A186A187A188A189A190A191A194A250A195A196A197A198KKHA761A2007A201A202A173A203A204A205A206D3A2075HT1AA209A210A211A212A213A214A215A216A217A218A219A220A221A222A223A215A224A225A226A227A212A228A229A230A231A232A233A234A235A236A237D3A209A210A238A239A240A241A242A243A238A239A240A244A245A223A246A231A232A247A248A241A249A252A253A254A255A2A227A59A0A143A1A233A8A255A232A32A338AA172A3A48BA178D3A13A5A6A7A172A9A10A55A126A56A57A11A92A12A14A61A15A96A16A17A18A19A6A62A231A63A12A80A20A55A173A64A21A22A23A24A66A257A26A27A28A299AA30KI18NMOLL1A31A34A35A68A36A37A38A39NGB2904A409BA41A42A69A105A70A191A43A44A45A46A47A48A105A71A49A50A42A51A73A52A53A54A58A147A42A60A65A67A72A7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